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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10611 | Brexpiprazole S-oxide D8 | DM-3411 D8 | Dopamine Receptor , 5-HT Receptor |
Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium labeled Brexpiprazole S-oxide. Brexpiprazole S-oxide is a main metabolite of Brexpiprazole. Brexpiprazole is a partial agonist of human 5-HT1A and dopamine receptors (... | |||
T10612 | Brexpiprazole S-oxide | DM-3411 | Dopamine Receptor , 5-HT Receptor |
Brexpiprazole S-oxide (DM-3411) is a main metabolite of Brexpiprazole. Brexpiprazole is a partial agonist of human 5-HT1A and dopamine receptors (Kis: 0.12 nM and 0.3 nM). |